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Apitolisib (GDC-0980)

Synonyms: (S)-1-(4-((2-(2-aminopyrimidin-5-yl)-7-methyl-4-morpholinothieno[3,2-d]pyrimidin-6-yl)methyl)piperazin-1-yl)-2-hydroxypropan-1-one
Cat. No.: A64400 CAS No.: 1032754-93-0
MDL.: Formula: C23H30N8O3S
F.W.498.6 Purity: 99%
Storage:
 
Size/Unit Price Qty Availability Price Total
5mg $120.00 Enter qty and click checkbox $120.00
Catalog Number: A64400   CAS No.: 1032754-93-0
MDL: Formula: C23H30N8O3S
F.W.: 498.6 Purity: 99%
Package: Unit: mg
Appearance: M.P.:
B.P.: Density:
Optical Rotation: Refractive Index:
Solubility: DMSO Stability:
Storage: Category: Reference Standard
Application: GDC-0980 (RG7422) is a selective, potent, orally bioavailable inhibitor of Class I PI3 kinase and mTOR kinase (TORC1/2) with in vitro IC50 of 5, 27, 7 and 14 nM for p110 a, ß, d and ? isoforms, respectively.