Catalog Number: |
Z78050 |
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CAS No.: |
1020720-04-0/68291-97-4(unlabelled) |
MDL: |
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Formula: |
C8H4D4N2O3S |
F.W.: |
216.25 |
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Purity: |
99% |
Package: |
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Unit: |
mg |
Appearance: |
Off-White to Light Brown Solid |
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M.P.: |
163-165°C |
B.P.: |
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Density: |
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Optical Rotation: |
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Refractive Index: |
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Solubility: |
DMSO (Slightly), Methanol (Slightly) |
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Stability: |
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Storage: |
-20°C Freezer, Under Inert Atmosphere |
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Category: |
Reference Standard |
Reference: |
Masuda, Y., et al.: Arzneim.-Forsch., 30, 477 (1980), Hammond, E.J., et al.: Gen. Pharmacol., 18, 303 (1987), Schmidt, D., et al.: Epilepsy Res., 15, 67 (1993), Sorkin, E.M., et al.: Drugs, 45, 760 (1993), |
Application: |
Labelled sulfonamide antiseizure agent; blocks repetitive firing of voltagesensitive sodium channels and reduces voltage-sensitive T-type calcium currents. Heterocyclic methanesulfonide with anticonvulsant properties. The compound is under investigation for potential therapeutic use as an antiepileptic drug. Anticonvulsant.
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Category: |
Aromatics, Isotope Labelled Compounds, Neurochemicals, Pharmaceuticals, Intermediates & Fine Chemicals, |